(3R,4R)-,2-HYDROXY-1,2,3-PROPANETRICARBOXYLATE(1:1);Xeljanz;CP-690550(Tofacitinibcitrate);(3R,4R)-1-(Cyanoacetyl)-4-methyl-N-methyl-N-1H-pyrrolo[2,3-d]pyrimidin-4-yl-3-piperidinamine2-hydroxy-1,2,3-palropanetricarboxylate
CAS:540737-29-9
CF: C16H20N6O.C6H8O7
MW:504.497
Availability: R&D; Commercialization
⬤ CAS No.540737-29-9
⬤ Packaging type：
20kg barrel；5kg barrel；1kg bag；500g bag ; Customized Packaging
| Product Name | Tofacitinib citrate |
| CAS No. | 540737-29-9 |
| Chemical Formula | C16H20N6O.C6H8O7 |
| Molecular Weight | 504.497 |
| Related Categories | Pharmaceutical raw materials; small molecule inhibitors; anticancer products; chemical reagents, fine chemicals, pharmaceutical intermediates, material intermediates; APIs |
| EINECS | 638-826-4 |
| Melting point | 201 °C (decomp) |
| Storage conditions | room temp |
| Solubility | Solubility in DMSO is 5 mg/mL (clear solution; heated) |
| Form | powder |
| Color | White to beige |
| Uses | Tofacitinib (477600-75-2) API is a Jak kinase inhibitor for the treatment of rheumatoid arthritis. |
| Adverse Reactions | In clinical trials, the most common adverse reactions of tofacitinib citrate were upper respiratory tract infection, headache, diarrhea, nasal congestion, sore throat and nasopharyngitis. |
| Note | This product is a chemical product and is only used for new drug research and development, process research, chemical intermediate reprocessing, etc. |
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